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Target Details
Name:
Alteplase
Uniprot name:
TPA_HUMAN
Accession Numbers:
A8K022
P00750
Q15103
Q503B0
Q6PJA5
Q7Z7N2
Q86YK8
Q9BU99
Q9BZW1
EC-Number:
3.4.21.68
Organism:
Homo sapiens
Human
PDB IDs:
1A5H
1BDA
1PK2
1PML
1RTF
1TPG
1TPK
1TPM
1TPN
KEGG Pathways:
show KEGG Pathways
Drugs:
Name
PubChem ID
Source
References
Interaction
1fax
122129
BindingDB
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show
1ghw
5326545
BindingDB
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show
1gi9
5326549
BindingDB
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show
1o2g
447476
BindingDB
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1o2h
447478
BindingDB
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1o3h
447508
BindingDB
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1o3p
5326663
BindingDB
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1owi
447734
BindingDB
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show
2-(2-hydroxyphenyl)-1H-indole-5-carboximidamide
1508
BindingDB
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2feq
23586156
BindingDB
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2jh5
9911502
BindingDB
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2uwo
10095865
BindingDB
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2uwp
10343728
BindingDB
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330942-05-7
10275777
BindingDB
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4-HYDROXY-3-[2-OXO-3-(THIENO[3,2-B]PYRIDINE-2-SULFONYLAMINO)-PYRROLIDIN-1-YLMETHYL]-BENZAMIDINE
5326514
BindingDB
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show
4-iodobenzo[b]thiophene-2-carboxamidine
1746
BindingDB
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4-[[1-methyl-5-[(2-methylbenzimidazol-1-yl)methyl]benzimidazol-2-yl]methylamino]benzenecarboximidamide
445756
BindingDB
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6-carbamimidoyl-N-phenylnaphthalene-2-carboxamide
447732
BindingDB
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show
6-CHLORO-2-(2-HYDROXY-BIPHENYL-3-YL)-1H-INDOLE-5-CARBOXAMIDINE
445843
BindingDB
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6-Chloro-2-(2-Hydroxybiphenyl-3-yl)-1H-Indole-5-Carboxamidine
445844
BindingDB
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show
6-FLUORO-2-(2-HYDROXY-3-ISOBUTOXY-PHENYL)-1H-BENZOIMIDAZOLE-5-CARBOXAMIDIN
5326553
BindingDB
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show
6-FLUORO-2-[2-HYDROXY-3-(2-METHYL-CYCLOHEXYLOXY)-PHENYL]-1H-INDOLE-5-CARBO
445849
BindingDB
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6-[N-(1-ISOPROPYL-3,4-DIHYDRO-7-ISOQUINOLINYL)CARBAMYL]-2-NAPHTHALENECARBOXAMIDINE
447735
BindingDB
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7-methoxy-8-(1-methylsulfonylpyrazol-4-yl)naphthalene-2-carboximidamide
5289529
BindingDB
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show
8-(PYRIMIDIN-2-YLAMINO)NAPHTHALENE-2-CARBOXIMIDAMIDE
448610
BindingDB
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show
Ac-Phe-pro-boroarg-OH
122296
BindingDB
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AC1L9GOC
444655
BindingDB
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AC1MPW2P
3392032
BindingDB
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AC1MV8RA
3729024
BindingDB
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AC1NS0VS
5326676
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AC1NS0WF
5326684
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AC1NS41B
5353305
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AC1O0UPY
6102526
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AC1O0UQP
6102594
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AC1O0UQS
6102595
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AC1O1DKC
6119062
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AC1O1DKF
6119063
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AC1OCEOE
6917805
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AIDS214692
10126451
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APC-10818
23646618
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APC-11417
23646620
BindingDB
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APC-9008
23646617
BindingDB
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APC-9850
23646621
BindingDB
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Benzenecarboximidamide
2332
BindingDB
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beta-Naphthamidine
193409
BindingDB
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BIBM1015
9953722
BindingDB
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BIBT0871
9600423
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CA-21
23644682
BindingDB
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CA-22
23646779
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CA-24
23646782
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CA-25
23646784
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CHEBI:646975
44347413
BindingDB
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CHEBI:651888
44347286
BindingDB
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CHEBI:652277
44366338
BindingDB
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CHEMBL101759
44330628
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CHEMBL102552
44335014
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CHEMBL104064
10116936
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CHEMBL104211
10225952
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CHEMBL104505
10278414
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CHEMBL104904
21707001
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CHEMBL105395
10294146
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CHEMBL105819
44338049
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CHEMBL107743
44335624
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CHEMBL107872
44339283
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CHEMBL107911
10648370
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CHEMBL108202
10529121
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CHEMBL1083499
9866964
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CHEMBL108447
9799627
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CHEMBL108717
10742217
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CHEMBL109274
44339119
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CHEMBL109287
11149953
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CHEMBL109535
11188793
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CHEMBL109751
21705171
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CHEMBL110358
44339233
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CHEMBL111036
44339192
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CHEMBL111338
11361949
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CHEMBL111432
11186243
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CHEMBL111471
11473486
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CHEMBL111543
11774107
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CHEMBL111567
11739438
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CHEMBL111660
11347670
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CHEMBL115982
10048688
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CHEMBL116136
44343561
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CHEMBL116137
10482360
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CHEMBL116405
44343829
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CHEMBL116406
44343830
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CHEMBL1172449
49798729
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CHEMBL117449
44343849
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CHEMBL117511
44343575
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CHEMBL117669
44343631
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CHEMBL117803
44343886
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CHEMBL122894
44347573
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CHEMBL125153
11824584
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CHEMBL126707
10959252
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CHEMBL127278
10871563
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CHEMBL127407
11782862
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CHEMBL127909
9884570
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CHEMBL135723
44356715
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CHEMBL138568
10505479
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CHEMBL138905
44359104
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CHEMBL139490
44358802
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CHEMBL139910
44358868
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CHEMBL139980
44358860
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CHEMBL140359
44359105
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CHEMBL141347
44359090
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CHEMBL141584
44359053
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CHEMBL141834
44359039
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CHEMBL148317
44367340
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CHEMBL151939
9915041
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CHEMBL153565
44367430
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CHEMBL154985
44367372
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CHEMBL159695
44376100
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CHEMBL162461
44376426
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CHEMBL163174
20641745
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CHEMBL172256
44386179
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CHEMBL172360
44385679
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CHEMBL172928
44383519
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CHEMBL173832
44386493
BindingDB
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CHEMBL174111
44386185
BindingDB
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CHEMBL174499
9959749
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CHEMBL174558
44386059
BindingDB
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CHEMBL174731
44385607
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CHEMBL174740
44385869
BindingDB
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CHEMBL174750
9959268
BindingDB
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CHEMBL174791
44385891
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CHEMBL174813
44385990
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CHEMBL174870
44386418
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CHEMBL174968
18727607
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CHEMBL175014
44386242
BindingDB
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CHEMBL175031
18727852
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CHEMBL175033
44385611
BindingDB
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CHEMBL175122
44385768
BindingDB
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CHEMBL175125
44386371
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CHEMBL175130
18727836
BindingDB
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CHEMBL175142
44386322
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CHEMBL175329
44385769
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CHEMBL176210
44387104
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CHEMBL176243
44386934
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CHEMBL176268
18727834
BindingDB
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CHEMBL176451
44385488
BindingDB
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CHEMBL176515
44385770
BindingDB
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CHEMBL176671
44385729
BindingDB
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CHEMBL176736
44385673
BindingDB
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CHEMBL176757
44385771
BindingDB
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CHEMBL176856
44386484
BindingDB
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CHEMBL177109
44385779
BindingDB
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CHEMBL177251
44386893
BindingDB
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CHEMBL177444
44387206
BindingDB
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CHEMBL177557
44385833
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CHEMBL177745
44386804
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CHEMBL181595
44392423
BindingDB
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CHEMBL181599
44392416
BindingDB
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CHEMBL182220
44392401
BindingDB
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CHEMBL182303
10216518
BindingDB
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CHEMBL182309
44392427
BindingDB
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CHEMBL182460
10287785
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CHEMBL182959
44392413
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CHEMBL183021
44392382
BindingDB
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CHEMBL185345
21707121
BindingDB
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CHEMBL18767
10054209
BindingDB
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CHEMBL189823
16086320
BindingDB
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CHEMBL194486
10024183
BindingDB
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CHEMBL194670
10052373
BindingDB
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CHEMBL197593
10051489
BindingDB
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CHEMBL197843
10390490
BindingDB
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CHEMBL198416
10003356
BindingDB
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CHEMBL198629
11720955
BindingDB
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CHEMBL198735
10390121
BindingDB
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CHEMBL198923
10409093
BindingDB
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CHEMBL198978
10324635
BindingDB
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CHEMBL205904
11948634
BindingDB
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CHEMBL20604
20595260
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CHEMBL206205
44411094
BindingDB
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CHEMBL20766
10007890
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CHEMBL207981
44411137
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CHEMBL208140
10479438
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CHEMBL20918
10389039
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CHEMBL20934
44274089
BindingDB
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CHEMBL21052
9803558
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CHEMBL21140
20595328
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CHEMBL213216
16086340
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CHEMBL214539
16086349
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CHEMBL214814
16086336
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CHEMBL215961
16086316
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CHEMBL221906
10297977
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CHEMBL224689
16658356
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CHEMBL226716
16658680
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CHEMBL227421
9952109
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CHEMBL227583
16658352
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CHEMBL227584
16658357
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CHEMBL227781
16658631
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CHEMBL227782
16658353
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CHEMBL227940
16658354
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CHEMBL233992
9954980
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CHEMBL236081
44433791
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CHEMBL237065
44434808
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CHEMBL237705
44434815
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CHEMBL238491
24750417
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CHEMBL238493
16718760
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CHEMBL238707
9827867
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CHEMBL238708
16718759
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CHEMBL238902
9912856
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CHEMBL238913
24748791
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CHEMBL239118
16718757
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CHEMBL239331
44436704
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CHEMBL239535
16718808
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CHEMBL239536
16718712
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CHEMBL239747
16718671
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CHEMBL263977
16086310
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CHEMBL264760
44303778
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CHEMBL265315
9910164
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CHEMBL277949
44274017
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CHEMBL27852
9850467
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CHEMBL279486
11755188
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CHEMBL281175
10391999
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CHEMBL282830
9937406
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CHEMBL284436
44278104
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CHEMBL287614
9956559
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CHEMBL28849
10472893
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CHEMBL289389
44286453
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CHEMBL291622
44304105
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CHEMBL29205
9822176
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CHEMBL292300
44303804
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CHEMBL292488
44304046
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CHEMBL292977
44303805
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CHEMBL293260
23646623
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CHEMBL293657
44303933
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CHEMBL294067
44303866
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CHEMBL294121
9805415
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CHEMBL294509
44303935
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CHEMBL294776
44304192
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CHEMBL297835
9826716
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CHEMBL300030
44298525
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CHEMBL302913
44303873
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CHEMBL303335
44303733
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CHEMBL303367
44303843
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44304097
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CHEMBL303978
44303854
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44303912
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CHEMBL305349
44303875
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CHEMBL306448
10391699
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CHEMBL316334
11068806
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CHEMBL316901
9807008
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CHEMBL317137
44330835
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CHEMBL317682
44330665
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CHEMBL318363
10903566
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CHEMBL318526
11824040
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CHEMBL318998
10074230
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44335601
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CHEMBL319047
10157296
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21707080
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CHEMBL31967
10248900
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44326715
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44334488
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9949275
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11244460
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21706943
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9804775
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10140847
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10185292
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10946869
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18771297
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10696955
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44339232
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44339270
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9935925
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44343885
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21192457
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44339231
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11782463
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44367355
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44367444
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44383242
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18727833
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10258264
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9871868
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10474680
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44392430
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44392405
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44392403
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44385772
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44386250
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44386366
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10027758
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44385541
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44385724
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44386622
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44386542
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10480463
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44386326
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44386637
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CHEMBL368494
44386891
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CHEMBL368614
18727831
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18727841
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44386642
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44387044
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44386841
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44386052
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44385935
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44386417
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44385998
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10074752
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10098302
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11419694
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9893177
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16086318
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16086308
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16086338
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16086312
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CHEMBL386249
16086344
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CHEMBL386275
16086342
BindingDB
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CHEMBL390310
16658633
BindingDB
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CHEMBL391344
16718762
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-
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CHEMBL391916
24748789
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CHEMBL391968
24749175
BindingDB
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CHEMBL391969
44436702
BindingDB
-
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CHEMBL392297
44434835
BindingDB
-
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CHEMBL393591
16049247
BindingDB
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CHEMBL393592
16718807
BindingDB
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CHEMBL393979
16718713
BindingDB
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CHEMBL394129
44434818
BindingDB
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CHEMBL39475
44286428
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CHEMBL398380
11237163
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CHEMBL399593
11351302
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CHEMBL40071
44286426
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CHEMBL401235
44434809
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CHEMBL403042
10275412
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CHEMBL404226
16086346
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CHEMBL405546
16086348
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CHEMBL411215
44416248
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CHEMBL412448
44303806
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CHEMBL41267
9890541
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CHEMBL415479
44264598
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CHEMBL416674
44303879
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CHEMBL417409
44303769
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CHEMBL418839
10432907
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CHEMBL418965
10302534
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CHEMBL419892
44330423
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CHEMBL420540
9871765
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CHEMBL421214
44334805
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CHEMBL423770
44367435
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CHEMBL423810
44376328
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CHEMBL42495
10669349
BindingDB
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CHEMBL425850
44386478
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CHEMBL425858
18727838
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CHEMBL425859
18727855
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CHEMBL426101
9954791
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CHEMBL426416
44386540
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CHEMBL426433
21707065
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CHEMBL431267
44325820
BindingDB
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CHEMBL431281
22883594
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CHEMBL431675
44347477
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CHEMBL432306
9954812
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CHEMBL433179
44326453
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CHEMBL433809
44386205
BindingDB
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CHEMBL435741
44385842
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CHEMBL436454
44380417
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CHEMBL437555
24180463
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CHEMBL439678
10067786
BindingDB
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CHEMBL44050
44290947
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CHEMBL441468
10744643
BindingDB
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CHEMBL442201
11292119
BindingDB
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CHEMBL444795
44343630
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CHEMBL447391
18727604
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CHEMBL450578
44432538
BindingDB
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CHEMBL472967
10205659
BindingDB
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CHEMBL479863
9808346
BindingDB
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CHEMBL48236
10255253
BindingDB
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CHEMBL487105
9935746
BindingDB
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CHEMBL49510
10480374
BindingDB
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CHEMBL515919
10298858
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CHEMBL52427
9949886
BindingDB
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CHEMBL53448
44298523
BindingDB
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CHEMBL53946
44298511
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CHEMBL54894
44298507
BindingDB
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CHEMBL55125
10131165
BindingDB
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CHEMBL55155
9948854
BindingDB
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CHEMBL55256
44298510
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CHEMBL553108
10390481
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CHEMBL55653
44298524
BindingDB
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CHEMBL569560
45485641
BindingDB
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CHEMBL569809
45485611
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CHEMBL570696
45485592
BindingDB
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CHEMBL571392
45485586
BindingDB
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CHEMBL571393
45485587
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CHEMBL571566
44626344
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CHEMBL571837
44626345
BindingDB
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CHEMBL571841
45485670
BindingDB
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CHEMBL572022
45485669
BindingDB
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CHEMBL572040
45485671
BindingDB
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CHEMBL572190
45485668
BindingDB
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CHEMBL572191
44626341
BindingDB
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CHEMBL572250
45485622
BindingDB
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CHEMBL579027
44626343
BindingDB
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CHEMBL583685
45485667
BindingDB
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CHEMBL593461
46196561
BindingDB
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CHEMBL593482
10324263
BindingDB
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CHEMBL59690
44304353
BindingDB
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CHEMBL59704
44303858
BindingDB
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CHEMBL59936
44304084
BindingDB
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CHEMBL60478
44304098
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CHEMBL60831
44303743
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CHEMBL61327
23646622
BindingDB
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CHEMBL61442
44303867
BindingDB
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CHEMBL61791
44303829
BindingDB
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CHEMBL62255
44303789
BindingDB
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CHEMBL62370
9884541
BindingDB
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CHEMBL62378
44303732
BindingDB
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CHEMBL62397
44303876
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CHEMBL62414
44303719
BindingDB
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CHEMBL62490
44303810
BindingDB
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CHEMBL62491
44303811
BindingDB
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CHEMBL62509
44303833
BindingDB
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CHEMBL62588
44303877
BindingDB
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CHEMBL62736
44303808
BindingDB
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CHEMBL62753
44303874
BindingDB
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CHEMBL63038
44303824
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CHEMBL63050
44304099
BindingDB
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CHEMBL63216
44303925
BindingDB
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CHEMBL64096
44303803
BindingDB
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CHEMBL64097
9886960
BindingDB
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CHEMBL64164
44304100
BindingDB
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CHEMBL64308
44304006
BindingDB
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CHEMBL64463
44303721
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CHEMBL64563
44304047
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CHEMBL64578
44304139
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CHEMBL64653
44304086
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CHEMBL64654
44304087
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CHEMBL64740
44304104
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CHEMBL64838
44303934
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CHEMBL64841
44303839
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CHEMBL67692
10001890
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CHEMBL6845
10521037
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CHEMBL69394
10347489
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CHEMBL70155
44311564
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CHEMBL70328
16678474
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CHEMBL70350
44311229
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CHEMBL7084
10624333
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CHEMBL71037
9802488
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CHEMBL72279
10367277
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CHEMBL7251
10648183
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CHEMBL7497
10765317
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CHEMBL7587
10345602
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CHEMBL7758
44264660
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CHEMBL7962
9913629
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CHEMBL80844
9987251
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CHEMBL85757
22883585
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CHEMBL90741
22883564
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CHEMBL91962
11015002
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CHEMBL92250
44326454
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CHEMBL92251
22556997
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CHEMBL92530
9911387
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CHEMBL92615
10144230
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CHEMBL92865
44325845
BindingDB
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CHEMBL92883
11057540
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CHEMBL92964
44325847
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CHEMBL93151
44325842
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CHEMBL93315
10075317
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CHEMBL93441
44326784
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CHEMBL93796
10574241
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CHEMBL94139
22557019
BindingDB
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CHEMBL94254
44326452
BindingDB
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CHEMBL94622
44327046
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CHEMBL94775
11057779
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CHEMBL94864
10303487
BindingDB
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CHEMBL94952
23004217
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CHEMBL95940
44330631
BindingDB
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CHEMBL95993
44330632
BindingDB
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CHEMBL96218
21967345
BindingDB
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CHEMBL96354
10302603
BindingDB
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CHEMBL96376
9984568
BindingDB
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CHEMBL96428
11089153
BindingDB
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CHEMBL96494
44326441
BindingDB
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CHEMBL96599
10185945
BindingDB
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CHEMBL96801
10143558
BindingDB
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CHEMBL96917
11009950
BindingDB
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CHEMBL98472
44330879
BindingDB
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CHEMBL98858
44331194
BindingDB
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CHEMBL99309
10026170
BindingDB
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CID 10311221
10624997
BindingDB
-
show
CID 10578280
10578280
BindingDB
-
show
CID 10790153
10367012
BindingDB
-
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CID 11200346
10200844
BindingDB
-
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CID 11247616
10181581
BindingDB
-
show
CID 11307837
11317532
BindingDB
-
show
CID 4713317
10816339
BindingDB
-
show
CID 5287492
10048823
BindingDB
-
show
CID 5326665
5326665
BindingDB
-
show
CID 5326669
5326669
BindingDB
-
show
CID 5326671
5326671
BindingDB
-
show
CID 5326671
5326696
BindingDB
-
show
CID 5326690
5326690
BindingDB
-
show
CID 9808035
9808035
BindingDB
-
show
CID 9823478
10717029
BindingDB
-
show
CID 9869156
9869156
BindingDB
-
show
CID 9895193
9895194
BindingDB
-
show
CID 9934590
9934590
BindingDB
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CID 9936104
10815545
BindingDB
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CID11010995
11010995
BindingDB
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CRA-10818
23646619
BindingDB
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show
cyanoguanidine, 3
44249821
BindingDB
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show
cyclic deriv. 33
9843775
BindingDB
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show
cyclic deriv. 34
16658181
BindingDB
-
show
cyclic deriv. 35
16658183
BindingDB
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show
cycloleucine deriv. 39
9956922
BindingDB
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show
cycloleucine deriv. 40
16658250
BindingDB
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show
cycloleucine deriv. 43
16658290
BindingDB
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cycloleucine deriv. 44
9956843
BindingDB
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cycloleucine deriv. 45
9935474
BindingDB
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show
Dabigatran
216210
BindingDB
-
show
efegatran
122267
BindingDB
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show
Epsilcapramine
564
DrugBank
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show
ESP
5438
BindingDB
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show
ESX
444753
BindingDB
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show
G17905
5326937
BindingDB
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Guanamprazine
16231
BindingDB
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Iloprost
6443959
DrugBank
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show
L86
5288687
BindingDB
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N-(1-ADAMANTYL)-N'-(4-GUANIDINOBENZYL)UREA
4286
BindingDB
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n-(4-carbamimidoyl-3-choro-phenyl)-2-hydroxy-3-iodo-5-methyl-benzamide
4300
BindingDB
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n-(4-carbamimidoyl-phenyl)-2-hydroxy-benzamide
4301
BindingDB
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N-[4-(aminomethyl)phenyl]-6-carbamimidoyl-4-(pyrimidin-2-ylamino)naphthalene-2-carboxamide
448605
BindingDB
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N-[4-(aminomethyl)phenyl]-6-carbamimidoylnaphthalene-2-carboxamide
447733
BindingDB
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Razaxaban
204102
BindingDB
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show
RPR120844
10322586
BindingDB
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show
substituted glycine deriv. 16
16658742
BindingDB
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show
substituted glycine deriv. 17
16658407
BindingDB
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show
substituted glycine deriv. 18
16658745
BindingDB
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show
substituted glycine deriv. 19
16658408
BindingDB
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show
substituted glycine deriv. 22
16657876
BindingDB
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show
substituted glycine deriv. 23
16657879
BindingDB
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show
substituted glycine deriv. 24
16657882
BindingDB
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substituted glycine deriv. 25
16657950
BindingDB
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show
substituted glycine deriv. 27
9930716
BindingDB
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show
substituted glycine deriv. 28
9822928
BindingDB
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show
substituted glycine deriv. 29
9802514
BindingDB
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show
substituted glycine deriv. 30
16658031
BindingDB
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show
Sulfonamidopyrrolidinone 20a
10790446
BindingDB
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show
TAK-442
11641515
BindingDB
-
show
Tranexamsaeure
5526
DrugBank
-
show
enlarge table
Synonyms:
Alteplase
Reteplase
t-PA
t-plasminogen activator
Tissue-type plasminogen activator
tPA
enlarge table
Similar targets:
Uniprot name
% Sequence similarity
% Sequence identity
B8ZX62_HUMAN
99.8
99.8
UROK_MOUSE
43.7
31.3
UROK_HUMAN
43
32.8
Q5PY49_HUMAN
42.4
32.6
THRB_MOUSE
37.3
26
FA9_HUMAN
36.4
25
THRB_BOVIN
36.2
25.6
FA10_HUMAN
35.9
24.3
THRB_HUMAN
34.9
25.4
PROC_HUMAN
34.5
23.4
FA11_HUMAN
34
23.2
FA7_HUMAN
33.9
23.5
FA10_BOVIN
33.2
24.9
CFAB_HUMAN
31.6
19
HGF_HUMAN
31.3
20.9
PROZ_HUMAN
31.2
19.7
MASP2_RAT
29.9
21.1
Q71SG6_HUMAN
29.6
18.6
PLMN_HUMAN
29.3
22
CHK1_YEAST
29.2
17.1
DEXT_PENMI
29.2
17.2
PAOX_HUMAN
29
17.9
HAO_NITEU
28.9
17.8
AMYB_HORVU
28.7
18.9
EXAA_PSEAE
28.4
17.3
C1S_HUMAN
28.2
18.5
DOPO_HUMAN
28.1
16.2
MDHP_FLABI
28.1
15.8
PP2BC_HUMAN
27.8
17
ASM_MOUSE
27.7
17.6
enlarge table
Protein-Protein Interactions:
Uniprot name
Source
UROK_HUMAN
PMID 16189514,7721771
TPA_HUMAN
2 PMIDs
TETN_HUMAN
3 PMIDs
NMDZ1_HUMAN
4 PMIDs
NEUS_HUMAN
5 PMIDs
LRP1_HUMAN
6 PMIDs
LRP1B_HUMAN
7 PMIDs
LAMA5_HUMAN
8 PMIDs
LAMA3_HUMAN
9 PMIDs
LAMA1_HUMAN
10 PMIDs
K2C8_HUMAN
11 PMIDs
IPSP_HUMAN
12 PMIDs
HMGB1_HUMAN
13 PMIDs
CKAP4_HUMAN
14 PMIDs
ANXA2_HUMAN
15 PMIDs
enlarge table
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