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Target Details
Name:
Peptidyl-prolyl cis-trans isomerase A
Uniprot name:
PPIA_HUMAN
Accession Numbers:
P05092
P62937
Q3KQW3
Q6IBU5
Q96IX3
Q9BRU4
Q9BTY9
Q9UC61
EC-Number:
5.2.1.8
Organism:
Homo sapiens
Human
PDB IDs:
1AK4
1AWQ
1AWR
1AWS
1AWT
1AWU
1AWV
1BCK
1CWA
1CWB
1CWC
1CWF
1CWH
1CWI
1CWJ
1CWK
1CWL
1CWM
1CWO
1FGL
1M63
1M9C
1M9D
1M9E
1M9F
1M9X
1M9Y
1MF8
1MIK
1NMK
1OCA
1RMH
1VBS
1VBT
1W8L
1W8M
1W8V
1YND
1ZKF
2ALF
2CPL
2CYH
2RMA
2RMB
3CYH
3CYS
4CYH
5CYH
KEGG Pathways:
-
Drugs:
Name
PubChem ID
Source
References
Interaction
()-oxazepam hemisuccinate sodium salt
44358264
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44358491
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44358265
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44358332
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44358492
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44358342
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
49863381
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
49863382
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
49863383
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
52946681
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
52940634
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
52945243
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
52946682
BindingDB
-
show
2-yl)benzenesulfonamide
44582823
BindingDB
-
show
AC1L9G81
444384
BindingDB
-
show
AC1LAX4R
497077
BindingDB
-
show
AC1LRDNV
1367020
BindingDB
-
show
AC1MUB56
3663276
BindingDB
-
show
AC1N4HBA
4128827
BindingDB
-
show
AC1N8XHV
4401642
BindingDB
-
show
AC1NN3AK
5020377
BindingDB
-
show
AC1NONRS
5116189
BindingDB
-
show
AI-204/31695004
11660364
BindingDB
-
show
AIDS085126
6475368
BindingDB
-
show
Bio-0872
16404350
BindingDB
-
show
Carboxypyrrolidine
145742
DrugBank
-
show
CHEBI:328305
9855081
BindingDB
-
show
CHEBI:328305
11643846
BindingDB
-
show
CHEMBL1269583
52941831
BindingDB
-
show
CHEMBL1269584
52947912
BindingDB
-
show
CHEMBL1269585
52946683
BindingDB
-
show
CHEMBL1269586
52945473
BindingDB
-
show
CHEMBL1269587
52947949
BindingDB
-
show
CHEMBL1269589
52940669
BindingDB
-
show
CHEMBL1269590
52940670
BindingDB
-
show
CHEMBL1269591
52940671
BindingDB
-
show
CHEMBL1269592
24814873
BindingDB
-
show
CHEMBL1269593
52945496
BindingDB
-
show
CHEMBL1269594
52947950
BindingDB
-
show
CHEMBL1269595
52941859
BindingDB
-
show
CHEMBL1269596
50899161
BindingDB
-
show
CHEMBL146970
44366403
BindingDB
-
show
CHEMBL148477
44366303
BindingDB
-
show
CHEMBL148546
44366208
BindingDB
-
show
CHEMBL148657
44366390
BindingDB
-
show
CHEMBL149224
44366350
BindingDB
-
show
CHEMBL150749
44366040
BindingDB
-
show
CHEMBL151360
44366261
BindingDB
-
show
CHEMBL151381
44366450
BindingDB
-
show
CHEMBL151384
44366232
BindingDB
-
show
CHEMBL151385
44366233
BindingDB
-
show
CHEMBL151816
44366260
BindingDB
-
show
CHEMBL198293
11717355
BindingDB
-
show
CHEMBL199550
11675245
BindingDB
-
show
CHEMBL201025
11531251
BindingDB
-
show
CHEMBL201113
11710570
BindingDB
-
show
CHEMBL201394
11639129
BindingDB
-
show
CHEMBL201395
11631957
BindingDB
-
show
CHEMBL201450
11638938
BindingDB
-
show
CHEMBL201645
11617502
BindingDB
-
show
CHEMBL201664
11588606
BindingDB
-
show
CHEMBL201718
11574097
BindingDB
-
show
CHEMBL203100
44406917
BindingDB
-
show
CHEMBL203142
11703833
BindingDB
-
show
CHEMBL203194
11516665
BindingDB
-
show
CHEMBL263062
44366453
BindingDB
-
show
CHEMBL264229
13037937
BindingDB
-
show
CHEMBL266308
44358399
BindingDB
-
show
CHEMBL266503
44358277
BindingDB
-
show
CHEMBL267710
44347614
BindingDB
-
show
CHEMBL274113
44358331
BindingDB
-
show
CHEMBL276363
44294709
BindingDB
-
show
CHEMBL295937
44294875
BindingDB
-
show
CHEMBL295942
44295258
BindingDB
-
show
CHEMBL296587
44294708
BindingDB
-
show
CHEMBL297131
44295050
BindingDB
-
show
CHEMBL299145
44295067
BindingDB
-
show
CHEMBL299202
44295153
BindingDB
-
show
CHEMBL299372
44295134
BindingDB
-
show
CHEMBL300089
44295136
BindingDB
-
show
CHEMBL300523
44294838
BindingDB
-
show
CHEMBL313327
10051106
BindingDB
-
show
CHEMBL314456
10023554
BindingDB
-
show
CHEMBL315033
11730110
BindingDB
-
show
CHEMBL329797
44321275
BindingDB
-
show
CHEMBL341860
44365970
BindingDB
-
show
CHEMBL356248
44366391
BindingDB
-
show
CHEMBL357384
44366144
BindingDB
-
show
CHEMBL358023
44366404
BindingDB
-
show
CHEMBL358478
44366351
BindingDB
-
show
CHEMBL358925
44366405
BindingDB
-
show
CHEMBL371213
11567780
BindingDB
-
show
CHEMBL373254
11632684
BindingDB
-
show
CHEMBL382465
11718015
BindingDB
-
show
CHEMBL382567
11559871
BindingDB
-
show
CHEMBL384058
44393427
BindingDB
-
show
CHEMBL384516
44358391
BindingDB
-
show
CHEMBL384718
44393512
BindingDB
-
show
CHEMBL384726
44341483
BindingDB
-
show
CHEMBL404789
44347622
BindingDB
-
show
CHEMBL405301
44358392
BindingDB
-
show
CHEMBL407342
44341642
BindingDB
-
show
CHEMBL407456
44393513
BindingDB
-
show
CHEMBL407798
44358330
BindingDB
-
show
CHEMBL408273
44358251
BindingDB
-
show
CHEMBL409139
44393426
BindingDB
-
show
CHEMBL409283
44358333
BindingDB
-
show
CHEMBL409911
44358288
BindingDB
-
show
CHEMBL413867
44393514
BindingDB
-
show
CHEMBL415597
44341507
BindingDB
-
show
CHEMBL424038
44295020
BindingDB
-
show
CHEMBL426517
44358250
BindingDB
-
show
CHEMBL433082
44294814
BindingDB
-
show
CHEMBL433738
44366452
BindingDB
-
show
CHEMBL434694
44366209
BindingDB
-
show
CHEMBL438817
44393425
BindingDB
-
show
CHEMBL439455
44358490
BindingDB
-
show
CHEMBL443992
25098030
BindingDB
-
show
CHEMBL445240
25098029
BindingDB
-
show
CHEMBL482839
44582699
BindingDB
-
show
CHEMBL482840
44582700
BindingDB
-
show
CHEMBL48778
44294978
BindingDB
-
show
CHEMBL48822
44294940
BindingDB
-
show
CHEMBL48825
44295056
BindingDB
-
show
CHEMBL48875
44294971
BindingDB
-
show
CHEMBL489001
44582756
BindingDB
-
show
CHEMBL489021
44582780
BindingDB
-
show
CHEMBL489042
44582824
BindingDB
-
show
CHEMBL489612
25097748
BindingDB
-
show
CHEMBL489614
25098028
BindingDB
-
show
CHEMBL490247
44582805
BindingDB
-
show
CHEMBL490840
20414882
BindingDB
-
show
CHEMBL490848
44582757
BindingDB
-
show
CHEMBL492070
25098032
BindingDB
-
show
CHEMBL49783
44294512
BindingDB
-
show
CHEMBL50531
44295152
BindingDB
-
show
CHEMBL50853
44294510
BindingDB
-
show
CHEMBL50854
44294511
BindingDB
-
show
CHEMBL50991
44294787
BindingDB
-
show
CHEMBL51248
44294970
BindingDB
-
show
CHEMBL51732
44295066
BindingDB
-
show
CHEMBL518980
44582698
BindingDB
-
show
CHEMBL52165
44294584
BindingDB
-
show
CHEMBL521943
42630203
BindingDB
-
show
CHEMBL522094
44582804
BindingDB
-
show
CHEMBL525897
44249040
BindingDB
-
show
CHEMBL540193
44366451
BindingDB
-
show
CHEMBL540479
44249303
BindingDB
-
show
CHEMBL549627
44248910
BindingDB
-
show
CHEMBL549755
44249309
BindingDB
-
show
CHEMBL550098
44249304
BindingDB
-
show
CHEMBL551508
44248913
BindingDB
-
show
CHEMBL551796
45269870
BindingDB
-
show
CHEMBL552181
44249307
BindingDB
-
show
CHEMBL552255
44249306
BindingDB
-
show
CHEMBL556893
44249310
BindingDB
-
show
CHEMBL557628
44248912
BindingDB
-
show
CHEMBL558302
44249174
BindingDB
-
show
CHEMBL559525
44249042
BindingDB
-
show
CHEMBL559858
44249305
BindingDB
-
show
CHEMBL560115
44249173
BindingDB
-
show
CHEMBL560173
44248911
BindingDB
-
show
CHEMBL560850
44249039
BindingDB
-
show
CHEMBL560851
44249041
BindingDB
-
show
CHEMBL564391
44248914
BindingDB
-
show
CHEMBL564539
44249170
BindingDB
-
show
CHEMBL564647
44249414
BindingDB
-
show
CHEMBL564826
44249044
BindingDB
-
show
CHEMBL569840
44249415
BindingDB
-
show
CHEMBL86442
11046232
BindingDB
-
show
CHEMBL86465
15293457
BindingDB
-
show
CHEMBL88028
10993110
BindingDB
-
show
CHEMBL89881
11091428
BindingDB
-
show
CID 10805065
10591196
BindingDB
-
show
CID 11833443
10891863
BindingDB
-
show
CID 11833443
11833443
BindingDB
-
show
cyclosporin A
5284373
BindingDB
-
show
cyclosporin A
5280754
BindingDB
-
show
CYCLOSPORINE
6435893
DrugBank
-
show
methoxyphenyl)benzenesulfonamide
19678899
BindingDB
-
show
methyl-L-valyl]
6476061
BindingDB
-
show
nitrophenyl)thiourea (D2)
20415061
BindingDB
-
show
Oprea1_029075
25047343
BindingDB
-
show
Oprea1_148017
25046022
BindingDB
-
show
Oprea1_179475
25044910
BindingDB
-
show
Oprea1_450954
13578706
BindingDB
-
show
Oprea1_643359
13578707
BindingDB
-
show
SCY-635
49863459
BindingDB
-
show
SCY-635
6479267
BindingDB
-
show
yl)benzenesulfonamide
13422114
BindingDB
-
show
ZINC00171159
2823177
BindingDB
-
show
ZINC00171166
2823184
BindingDB
-
show
ZINC00171175
2823189
BindingDB
-
show
enlarge table
Synonyms:
Cyclophilin A
Cyclosporin A-binding protein
Peptidyl-prolyl cis-trans isomerase A
PPIase A
Rotamase A
enlarge table
Similar targets:
Uniprot name
% Sequence similarity
% Sequence identity
PPIA_PAPAN
100
100
PPIF_HUMAN
67.1
59.9
PPIH_HUMAN
65.7
51.1
PPIB_HUMAN
57.6
49.3
CYP5_CAEEL
56.4
46.6
PPIC_HUMAN
52.3
44.4
SAT2_HUMAN
38.7
20.9
MYG_PIG
33.7
21.6
RISB_AQUAE
33.5
17.3
CYC2_RHOVI
33.1
21.1
CANB1_HUMAN
32.5
19.8
SODC_BOVIN
32.4
21.8
SAV_STRAV
32.2
19.7
Q9X9L0_THETH
32.2
18.8
AZRB_BACOY
31.9
18.6
FUCL_ANGAN
31.6
16.6
ICYA_MANSE
31.5
19.6
MACM_STRMA
31.5
20.7
PHI_METJA
31
18.7
ARF2_YEAST
30.8
17.5
RL13_DEIRA
30.7
16.3
MYG_HORSE
30.6
22.8
ACPS_BACSU
30.6
17.3
CBIT_METTH
30.5
18.3
NIKR_SHIFL
30.5
17.5
SODC_SCHMA
30.4
21.5
Y1796_ARCFU
30.2
17.5
Q9RW27_DEIRA
30.2
18
GLB1_SCAIN
30.2
17.7
GSTP_ONCVO
30
16
enlarge table
Protein-Protein Interactions:
Uniprot name
Source
UNG_HUMAN
PMID 16049941
UCHL1_HUMAN
2 PMIDs
UCHL1_HUMAN
3 PMIDs
TYY1_HUMAN
4 PMIDs
TBB5_HUMAN
5 PMIDs
TBB5_HUMAN
6 PMIDs
STXB1_HUMAN
7 PMIDs
SPTA2_HUMAN
8 PMIDs
SPT5H_HUMAN
9 PMIDs
S10A8_HUMAN
10 PMIDs
Q71V99_HUMAN
11 PMIDs
PTPRN_HUMAN
12 PMIDs
PSIP1_HUMAN
13 PMIDs
PRS23_HUMAN
14 PMIDs
PRR13_HUMAN
15 PMIDs
PRLR_HUMAN
16 PMIDs
PPIA_HUMAN
17 PMIDs
PP2BA_HUMAN
18 PMIDs
PGAM1_HUMAN
19 PMIDs
PGAM1_HUMAN
20 PMIDs
NSF_HUMAN
21 PMIDs
NSF_HUMAN
22 PMIDs
NFL_HUMAN
23 PMIDs
NFL_HUMAN
24 PMIDs
MBP_HUMAN
25 PMIDs
M3K5_HUMAN
26 PMIDs
M3K5_HUMAN
27 PMIDs
JAK2_HUMAN
28 PMIDs
ITK_HUMAN
29 PMIDs
HSP7C_HUMAN
30 PMIDs
HSP7C_HUMAN
31 PMIDs
HS90A_HUMAN
32 PMIDs
HS90A_HUMAN
33 PMIDs
HMGA1_HUMAN
34 PMIDs
GRB2_HUMAN
35 PMIDs
GFAP_HUMAN
36 PMIDs
GFAP_HUMAN
37 PMIDs
DYN1_HUMAN
38 PMIDs
DYN1_HUMAN
39 PMIDs
DYH1_HUMAN
40 PMIDs
CXCR4_HUMAN
41 PMIDs
CRYAB_HUMAN
42 PMIDs
CRYAB_HUMAN
43 PMIDs
CD99_HUMAN
44 PMIDs
CD4_HUMAN
45 PMIDs
CCR5_HUMAN
46 PMIDs
CANB1_HUMAN
47 PMIDs
BAF_HUMAN
48 PMIDs
APBB1_HUMAN
49 PMIDs
ACTB_HUMAN
50 PMIDs
ACTB_HUMAN
51 PMIDs
ABC3G_HUMAN
52 PMIDs
A4_HUMAN
53 PMIDs
A4_HUMAN
54 PMIDs
A4_HUMAN
55 PMIDs
1433Z_HUMAN
56 PMIDs
1433Z_HUMAN
57 PMIDs
1433Z_HUMAN
58 PMIDs
enlarge table
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