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Target Details
Name:
cAMP-dependent protein kinase catalytic subunit alpha
Uniprot name:
KAPCA_MOUSE
Accession Numbers:
P05132
Q9JID0
EC-Number:
2.7.11.11
Organism:
Mouse
Mus musculus
PDB IDs:
1APM
1ATP
1BKX
1BX6
1FMO
1J3H
1JBP
1JLU
1L3R
1PVK
1RDQ
1RE8
1REJ
1REK
1SYK
2CPK
2ERZ
2QCS
2QUR
2QVS
3FHI
3FJQ
KEGG Pathways:
show KEGG Pathways
Drugs:
Name
PubChem ID
Source
References
Interaction
()-oxazepam hemisuccinate sodium salt
25190768
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
25190769
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
25190790
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
16121514
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
25190791
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44282246
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44282442
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44282443
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44282377
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44282232
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44282376
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44282430
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44282245
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44282233
BindingDB
-
show
()-oxazepam hemisuccinate sodium salt
44282230
BindingDB
-
show
(S)-2-METHYL-1-[(4-METHYL-5-ISOQUINOLINE)SULFONYL]-HOMOPIPERAZINE
448043
BindingDB
-
show
2-METHYL-2,4-PENTANEDIOL
5288834
DrugBank
-
show
Arabinosyladenine
191
BindingDB
-
show
BALANOL
5287736
DrugBank
-
show
Balanol analog 2
5327919
DrugBank
-
show
BALANOL ANALOG 8
448327
DrugBank
-
show
CHEBI:148314
44282203
BindingDB
-
show
CHEBI:148350
44282231
BindingDB
-
show
CHEMBL178945
10185160
BindingDB
-
show
CHEMBL297394
25190767
BindingDB
-
show
CHEMBL359486
10302405
BindingDB
-
show
CHEMBL360304
10143584
BindingDB
-
show
CHEMBL368416
10163439
BindingDB
-
show
CHEMBL368895
10209082
BindingDB
-
show
CHEMBL426587
10187378
BindingDB
-
show
CHEMBL447678
25190789
BindingDB
-
show
CHEMBL449834
25190785
BindingDB
-
show
CHEMBL450179
25141061
BindingDB
-
show
CHEMBL450260
25190781
BindingDB
-
show
CHEMBL454225
25190782
BindingDB
-
show
CHEMBL465518
25190786
BindingDB
-
show
CHEMBL495088
25190784
BindingDB
-
show
CHEMBL495766
25190765
BindingDB
-
show
CHEMBL495767
25190773
BindingDB
-
show
CHEMBL496141
25190778
BindingDB
-
show
CHEMBL496365
25190772
BindingDB
-
show
CHEMBL497800
25190777
BindingDB
-
show
CHEMBL498924
25190771
BindingDB
-
show
CHEMBL500989
25190783
BindingDB
-
show
CHEMBL501706
25190766
BindingDB
-
show
CHEMBL505949
25190770
BindingDB
-
show
CHEMBL506331
25190788
BindingDB
-
show
CHEMBL509411
25190787
BindingDB
-
show
CHEMBL510221
25190779
BindingDB
-
show
CHEMBL521551
25190774
BindingDB
-
show
CHEMBL522899
25190780
BindingDB
-
show
CHEMBL523401
25190776
BindingDB
-
show
CHEMBL523738
25190775
BindingDB
-
show
Fasudil hydrochloride
3547
BindingDB
-
show
HYDROXYFASUDIL
3064778
BindingDB
-
show
HYDROXYFASUDIL
3064778
DrugBank
-
show
L-Cysteine, mercaptoethanol mixed disulfide
170018
DrugBank
-
show
Methylheptane
356
DrugBank
-
show
N-(2-(4-Bromocinnamylamino)ethyl)-5-isoquinolinesulfonamide
449241
BindingDB
-
show
N-(2-(4-Bromocinnamylamino)ethyl)-5-isoquinolinesulfonamide
449241
PROMISCUOUS
PMID 15062850
show
nchembio.95-comp18
3501
PROMISCUOUS
PMID 16248886
show
Phosphatidalserine
68841
DrugBank
-
show
PHOSPHONOTHREONINE
3246323
DrugBank
-
show
STAUROSPORINE
44259
BindingDB
-
show
staurosporine
44299148
BindingDB
-
show
Succinonitrile, bis(amino(o-aminophenylthio)methylene)-
3006531
PROMISCUOUS
PMID 11640885
show
Tetrahydrocannabinols
2977
PROMISCUOUS
PMID 9260875
show
Tetrahydrocannabinols
16078
PROMISCUOUS
PMID 9260875
show
Valerylaldehyde
8063
DrugBank
-
show
Vidarabine
6713976
BindingDB
-
show
y-27632
448042
BindingDB
-
show
enlarge table
Synonyms:
cAMP-dependent protein kinase catalytic subunit alpha
PKA C-alpha
enlarge table
Similar targets:
Uniprot name
% Sequence similarity
% Sequence identity
KAPCA_HUMAN
99.4
98
KAPCA_RAT
99.1
99.1
KAPCA_PIG
99.1
97.4
KAPCA_BOVIN
98.9
97.7
KAPCB_HUMAN
95.2
92
KAPCB_MOUSE
94.3
91.5
KAPCB_RAT
94.3
91.5
KAPCG_HUMAN
91.5
81.5
KAPA_YEAST
60.1
40.6
MK14_MOUSE
43
20.4
MK14_HUMAN
42.7
20.4
AKT1_MOUSE
42.7
28.7
AKT1_HUMAN
42.5
28.5
MAPK2_HUMAN
41.1
24.1
MK12_HUMAN
40.3
20.5
MAPK2_CRILO
39.9
24
MK01_HUMAN
39.1
22.4
MK01_MOUSE
39.1
22.5
MK01_RAT
39.1
22.5
Q1HBJ4_HUMAN
39.1
22.4
Q499G7_HUMAN
38.6
22.2
MP2K2_HUMAN
37.5
20.8
MP2K3_MOUSE
37.4
22.1
CDK9_HUMAN
37.4
19.4
MK03_RAT
37.1
21.7
MK03_MOUSE
37.1
21.7
MP2K2_MOUSE
37
19.8
MP2K6_MOUSE
36.7
21.7
STK6_HUMAN
36.4
21.3
PIM1_FELCA
36.4
21.4
enlarge table
Protein-Protein Interactions:
No data available
enlarge table
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