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Target Details
Name:
Glutamate receptor 2
Uniprot name:
GRIA2_RAT
Accession Numbers:
P19491
Q9R174
EC-Number:
-
Organism:
Rat
Rattus norvegicus
PDB IDs:
1FTJ
1FTK
1FTL
1FTM
1FTO
1FW0
1GR2
1LB8
1LB9
1LBB
1LBC
1M5B
1M5C
1M5D
1M5E
1M5F
1MM6
1MM7
1MQD
1MQG
1MQH
1MQI
1MQJ
1MS7
1MXU
1MXV
1MXW
1MXX
1MXY
1MXZ
1MY0
1MY1
1MY2
1MY3
1MY4
1N0T
1NNK
1NNP
1P1N
1P1O
1P1Q
1P1U
1P1W
1SYH
1SYI
1WVJ
1XHY
2AIX
2AL4
2AL5
2ANJ
2CMO
2GFE
2I3V
2I3W
2P2A
2UXA
3B6Q
3B6T
3B6W
3B7D
3BBR
3BFT
3BFU
3BKI
3DP6
3H03
3H06
3H5V
3H5W
3H6T
3H6U
3H6V
3H6W
3IJO
3IJX
3IK6
3IL1
3ILT
3ILU
KEGG Pathways:
show KEGG Pathways
Drugs:
Name
PubChem ID
Source
References
Interaction
(S)-DES-ME-AMPA
447195
DrugBank
-
show
14598502
14598502
BindingDB
-
show
1nnk
447407
BindingDB
-
show
2-AMINO-3-(3-HYDROXY-7,8-DIHYDRO-6H-CYCLOHEPTA[D]-4-ISOXAZOLYL)PROPIONIC ACID
5288598
BindingDB
-
show
2-AMINO-3-(3-HYDROXY-7,8-DIHYDRO-6H-CYCLOHEPTA[D]-4-ISOXAZOLYL)PROPIONIC ACID
5288598
DrugBank
-
show
2-AMINO-3-(5-TERT-BUTYL-3-(PHOSPHONOMETHOXY)-4-ISOXAZOLYL)PROPIONIC ACID
447249
DrugBank
-
show
3-(5-Chloro-2,4-Dioxo-3,4-Dihydropyrimidin-1(2h)-Yl)-L-Alanine
44152410
BindingDB
-
show
3-(5-TERT-BUTYL-3-OXIDOISOXAZOL-4-YL)-L-ALANINATE
5287901
DrugBank
-
show
6,7-Dinitroquinoxaline-2,3-dione
3899541
DrugBank
-
show
71366-32-0
2733518
BindingDB
-
show
AC1MRQ5R
3496893
BindingDB
-
show
AC1NG5HR
4694356
BindingDB
-
show
ampa
1221
BindingDB
-
show
ANIRACETAM
2196
DrugBank
-
show
ANIRACETAM
2196
SuperTarget
-
show
BN1
447081
BindingDB
-
show
BROMO-WILLARDIINE
167842
DrugBank
-
show
CHEMBL1094129
46237944
BindingDB
-
show
CHEMBL1098101
46238075
BindingDB
-
show
CHEMBL1098104
46238077
BindingDB
-
show
CHEMBL154700
9799478
BindingDB
-
show
CHEMBL193087
11818375
BindingDB
-
show
CHEMBL224688
9977288
BindingDB
-
show
CHEMBL224872
11742032
BindingDB
-
show
CHEMBL224926
10091990
BindingDB
-
show
CHEMBL346524
10132082
BindingDB
-
show
CHEMBL370941
11288627
BindingDB
-
show
CHEMBL372643
11219775
BindingDB
-
show
CHEMBL387549
10409259
BindingDB
-
show
CHEMBL388746
16659202
BindingDB
-
show
CHEMBL492469
24755637
BindingDB
-
show
CHEMBL492628
25129888
BindingDB
-
show
CHEMBL492629
24850231
BindingDB
-
show
CHEMBL492630
24850230
BindingDB
-
show
CHEMBL493596
25130238
BindingDB
-
show
CHEMBL493665
25129887
BindingDB
-
show
CHEMBL493892
25129891
BindingDB
-
show
CHEMBL508818
25129889
BindingDB
-
show
CHEMBL553028
44222306
BindingDB
-
show
CYCLOTHIAZIDE
2910
BindingDB
-
show
CYCLOTHIAZIDE
2910
DrugBank
-
show
CYCLOTHIAZIDE
5388988
DrugBank
-
show
CYCLOTHIAZIDE
2910
SuperTarget
-
show
CYCLOTHIAZIDE
5388988
SuperTarget
-
show
D-Glutaminsaeure
23327
BindingDB
-
show
DB03240
657004
BindingDB
-
show
DB03240
657004
DrugBank
-
show
Digensaeure
10255
BindingDB
-
show
DL-Willardiine
5123
BindingDB
-
show
Essigsaeure
176
DrugBank
-
show
FLUORO-WILLARDIINE
126569
BindingDB
-
show
FLUORO-WILLARDIINE
126569
DrugBank
-
show
Glutamicol
33032
BindingDB
-
show
IODO-WILLARDIINE
447196
BindingDB
-
show
IODO-WILLARDIINE
447196
DrugBank
-
show
Phosphaglycine
14017
DrugBank
-
show
Quisqualate
40539
DrugBank
-
show
THIO-ATPA
5289518
DrugBank
-
show
UBC
6420161
BindingDB
-
show
Willardiine
440053
DrugBank
-
show
enlarge table
Synonyms:
AMPA-selective glutamate receptor 2
GluR-2
GluR-B
GluR-K2
Glutamate receptor 2
Glutamate receptor ionotropic, AMPA 2
enlarge table
Similar targets:
Uniprot name
% Sequence similarity
% Sequence identity
GRIA2_HUMAN
99.5
99.5
Q59F93_HUMAN
95.8
95.4
GRIA3_HUMAN
85.6
71.7
GRIA4_HUMAN
81.2
68.2
GRIA1_HUMAN
79.1
66.1
GRIK1_HUMAN
55
36.7
GRIK2_HUMAN
54.7
37
GRIK3_HUMAN
54.5
36.9
GRIK2_RAT
54.5
36.7
GRIK4_HUMAN
48.6
32.3
GRIK5_HUMAN
47.2
31.3
GRID2_HUMAN
43.2
24.3
GRID1_HUMAN
41.2
25.1
Q5VSF4_HUMAN
41.1
23.5
Q9UPF9_HUMAN
41.1
23.4
Q5VSF9_HUMAN
40.6
22.9
Q5VSF5_HUMAN
40.2
22.8
Q9UPF8_HUMAN
40.2
22.7
NMDZ1_HUMAN
39.8
23
NMDZ1_RAT
39.4
23.1
Q59H41_HUMAN
39.4
22.8
NMD3B_HUMAN
33.4
19.5
NMD3A_RAT
32.6
18
NMD3A_HUMAN
31.8
17.8
OGA_CLOPE
31
16.9
VCAM1_HUMAN
30.8
16.3
GUC2C_PIG
30.6
17.5
KINH_HUMAN
30.6
17.4
RIR1_HUMAN
30.3
16.8
PDE6A_BOVIN
29.9
17.1
enlarge table
Protein-Protein Interactions:
No data available
enlarge table
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