SuperToxic
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Information
Structure
Synonyms:
119673-08-4
5H-Indolo[2,3-a]pyrrolo[3,4-c]carbazole-5,7 (6H)-dione, 1, 11-.beta.-D-glucopyranosyl)-
BMS-181176
BMY 27557
NSC655649
Rebeccamycin analog
Smile:
c1cc2c(c(c1)Cl)n(c1c2c2c(c3c4c(c(ccc4)Cl)[nH]c13)c(=O)n(c2=O)CCN(CC)CC)[C@@H]1O[C@H]([C@H]([C@H]([C@H]1O)O)OC)CO
Cas:
119673-08-4
NSC:
640199
Formula:
C33H34Cl2N4O7
Rings:
7
Atoms:
80
Weight:
669.552
H-Donors:
4
H-Acceptor:
10
Rotatable Bonds:
8
NCI-H226
4 nlog(LC50)
Cellline
Tox Value
Tox Type
Cellline
Tox Value
Tox Type
Cellline
Tox Value
Tox Type
NCI-H226
4
nlog(LC50)
OVCAR-5
4
nlog(LC50)
CCRF-CEM
4
nlog(LC50)
MOLT-4
4
nlog(LC50)
HT29
4
nlog(LC50)
COLO 205
4
nlog(LC50)
HCT-15
4
nlog(LC50)
Hs 578T
4
nlog(LC50)
T-47D
4
nlog(LC50)
SK-OV-3
4
nlog(LC50)
MOLT-4
4
nlog(LC50)
HL-60(TB)
4
nlog(LC50)
SR
4
nlog(LC50)
SN12C
4
nlog(LC50)
LOX IMVI
4
nlog(LC50)
SNB-19
4
nlog(LC50)
SNB-75
4
nlog(LC50)
U251
4
nlog(LC50)
K-562
4.253
nlog(LC50)
IGROV1
4.295
nlog(LC50)
TK-10
4.584
nlog(LC50)
RPMI-8226
4.655
nlog(LC50)
ACHN
4.655
nlog(LC50)
SNB-19
4.692
nlog(LC50)
HOP-18
4.702
nlog(LC50)
HCT-15
4.74
nlog(LC50)
COLO 205
4.766
nlog(LC50)
MCF7
4.773
nlog(LC50)
CAKI-1
4.779
nlog(LC50)
SF-268
4.783
nlog(LC50)
OVCAR-8
4.847
nlog(LC50)
NCI-H460
4.915
nlog(LC50)
DU-145
5.006
nlog(LC50)
EKVX
5.019
nlog(LC50)
KM20L2
5.051
nlog(LC50)
PC-3
5.059
nlog(LC50)
A549/ATCC
5.062
nlog(LC50)
OVCAR-3
5.074
nlog(LC50)
SK-MEL-2
5.091
nlog(LC50)
HOP-92
5.111
nlog(LC50)
CAKI-1
5.131
nlog(LC50)
SW-620
5.135
nlog(LC50)
NCI-H522
5.149
nlog(LC50)
UACC-257
5.161
nlog(LC50)
IGROV1
5.167
nlog(LC50)
DLD-1
5.17
nlog(LC50)
SNB-78
5.227
nlog(LC50)
SK-OV-3
5.252
nlog(LC50)
DMS 114
5.258
nlog(LC50)
SF-295
5.264
nlog(LC50)
HL-60(TB)
5.272
nlog(LC50)
OVCAR-4
5.293
nlog(LC50)
BT-549
5.314
nlog(LC50)
EKVX
5.337
nlog(LC50)
NCI-H322M
5.354
nlog(LC50)
OVCAR-5
5.369
nlog(LC50)
OVCAR-3
5.409
nlog(LC50)
SK-MEL-28
5.413
nlog(LC50)
HCT-116
5.42
nlog(LC50)
MDA-MB-231/ATCC
5.425
nlog(LC50)
KM12
5.451
nlog(LC50)
SK-MEL-28
5.465
nlog(LC50)
M19-MEL
5.466
nlog(LC50)
HT29
5.468
nlog(LC50)
NCI-H322M
5.472
nlog(LC50)
KM12
5.476
nlog(LC50)
UACC-257
5.476
nlog(LC50)
SN12C
5.486
nlog(LC50)
Malme-3M
5.491
nlog(LC50)
786-0
5.502
nlog(LC50)
786-0
5.517
nlog(LC50)
OVCAR-4
5.538
nlog(LC50)
NCI-H460
5.549
nlog(LC50)
SK-MEL-5
5.557
nlog(LC50)
U251
5.568
nlog(LC50)
HOP-62
5.568
nlog(LC50)
DMS 273
5.617
nlog(LC50)
SNB-75
5.626
nlog(LC50)
HOP-92
5.636
nlog(LC50)
SF-295
5.64
nlog(LC50)
A549/ATCC
5.643
nlog(LC50)
RXF-631
5.653
nlog(LC50)
UO-31
5.671
nlog(LC50)
TK-10
5.673
nlog(LC50)
SR
5.69
nlog(LC50)
SW-620
5.704
nlog(LC50)
ACHN
5.708
nlog(LC50)
LXFL 529
5.73
nlog(LC50)
NCI-H226
5.756
nlog(LC50)
SF-539
5.813
nlog(LC50)
XF 498
5.813
nlog(LC50)
UO-31
5.877
nlog(LC50)
HCT-116
5.893
nlog(LC50)
SK-MEL-2
5.897
nlog(LC50)
HOP-62
5.964
nlog(LC50)
HCC-2998
5.974
nlog(LC50)
M14
5.986
nlog(LC50)
CCRF-CEM
6
nlog(LC50)
SR
6
nlog(LC50)
A498
6.033
nlog(LC50)
UACC-62
6.038
nlog(LC50)
RXF 393
6.053
nlog(LC50)
SK-MEL-5
6.061
nlog(LC50)
Malme-3M
6.08
nlog(LC50)
MDA-MB-435
6.115
nlog(LC50)
NCI-H23
6.123
nlog(LC50)
A498
6.141
nlog(LC50)
UACC-62
6.143
nlog(LC50)
M14
6.152
nlog(LC50)
MDA-N
6.157
nlog(LC50)
NCI-H522
6.221
nlog(LC50)
NCI-H23
6.248
nlog(LC50)
RPMI-8226
6.304
nlog(LC50)
RXF 393
6.321
nlog(LC50)
HCC-2998
6.472
nlog(LC50)
SF-539
6.539
nlog(LC50)
MOLT-4
6.718
nlog(LC50)
K-562
6.789
nlog(LC50)
LOX IMVI
6.83
nlog(LC50)
HT29
7.084
nlog(LC50)
OVCAR-5
7.142
nlog(LC50)
TK-10
7.145
nlog(LC50)
SNB-78
7.222
nlog(LC50)
DLD-1
7.316
nlog(LC50)
NCI-H322M
7.363
nlog(LC50)
U251
7.394
nlog(LC50)
UACC-257
7.424
nlog(LC50)
HOP-18
7.453
nlog(LC50)
KM20L2
7.461
nlog(LC50)
HCT-15
7.464
nlog(LC50)
HOP-92
7.484
nlog(LC50)
SF-295
7.485
nlog(LC50)
SK-MEL-28
7.504
nlog(LC50)
SF-268
7.507
nlog(LC50)
786-0
7.51
nlog(LC50)
ACHN
7.538
nlog(LC50)
SN12C
7.543
nlog(LC50)
SK-OV-3
7.572
nlog(LC50)
KM12
7.573
nlog(LC50)
OVCAR-8
7.581
nlog(LC50)
SW-620
7.623
nlog(LC50)
SNB-75
7.624
nlog(LC50)
LXFL 529
7.63
nlog(LC50)
NCI-H460
7.653
nlog(LC50)
OVCAR-3
7.728
nlog(LC50)
Malme-3M
7.739
nlog(LC50)
EKVX
7.741
nlog(LC50)
SK-MEL-5
7.751
nlog(LC50)
LOX IMVI
7.757
nlog(LC50)
CAKI-1
7.767
nlog(LC50)
NCI-H226
7.773
nlog(LC50)
M14
7.786
nlog(LC50)
HOP-62
7.791
nlog(LC50)
HCT-116
7.8
nlog(LC50)
SF-539
7.804
nlog(LC50)
SNB-19
7.889
nlog(LC50)
UO-31
7.921
nlog(LC50)
OVCAR-4
7.94
nlog(LC50)
NCI-H23
7.962
nlog(LC50)
IGROV1
8.019
nlog(LC50)
SK-MEL-2
8.117
nlog(LC50)
A498
8.121
nlog(LC50)
COLO 205
8.266
nlog(LC50)
DMS 273
8.283
nlog(LC50)
M19-MEL
8.309
nlog(LC50)
DMS 114
8.31
nlog(LC50)
HCC-2998
8.325
nlog(LC50)
A549/ATCC
8.352
nlog(LC50)
RXF 393
8.498
nlog(LC50)
UACC-62
8.656
nlog(LC50)